Chemicals and Drugs

Celiprolol

A cardioselective beta-1 adrenergic antagonist that has intrinsic sympathomimetic activity. It is used in the management of ANGINA PECTORIS and HYPERTENSION.

National Library of MedicineMedical Subject Headings2026

Structured Summary

Abstract

A cardioselective beta-1 adrenergic antagonist that has intrinsic sympathomimetic activity. It is used in the management of ANGINA PECTORIS and HYPERTENSION.

Chemical Identity

Chemical Information

Molecular Formula
C20H33N3O4
Molecular Weight
379.5 g/mol
CAS Registry No.
56980-93-9
IUPAC Name
3-[3-acetyl-4-[3-(tert-butylamino)-2-hydroxypropoxy]phenyl]-1,1-diethylurea
InChIKey
JOATXPAWOHTVSZ-UHFFFAOYSA-N
SMILES
CCN(CC)C(=O)NC1=CC(=C(C=C1)OCC(CNC(C)(C)C)O)C(=O)C
MeSH Unique ID
D017272
Source
PubChem CID 2663

MeSH Record

Classification

Broader headings

Related Concepts

Knowledge Graph

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Drug Class

Pharmacological Action

MeSH Record

Synonyms

17 entry terms
  • N'-(3-Acetyl-4-(3-((1,1-dimethylethyl)amino)-2-hydroxypropoxy)phenyl)-N,N-diethylurea
  • Celiprolol Hydrochloride
  • Celiprolol Monohydrochloride
  • Celiprolol, (+,-)-Isomer
  • Celiprolol, (R)-Isomer
  • Celiprolol, (S)-Isomer
  • Celiprolol, Monohydrochloride, (R)-Isomer
  • Celiprolol, Monohydrochloride, (S)-Isomer
  • REV-5320A
  • ST-1396
  • Selectol
  • Hydrochloride, Celiprolol
  • Monohydrochloride, Celiprolol
  • REV 5320A
  • REV5320A
  • ST 1396
  • ST1396

MeSH Record

Aspects Covered

25 allowable subheadings

Indexed with the subheadings administration & dosage, adverse effects, agonists, analogs & derivatives, analysis, antagonists & inhibitors, blood, cerebrospinal fluid, chemical synthesis, chemistry, classification, economics, history, immunology, isolation & purification, metabolism, pharmacokinetics, pharmacology, poisoning, radiation effects, standards, supply & distribution, therapeutic use, toxicity, urine.

MeSH Record

History Note

93; was CELIPROLOL (NM) 1978-92

MeSH Record

Previous Indexing

  • Propanolamines (1982-1992)
  • Urea/analogs & derivatives (1978-1982)

MeSH Hierarchy

Tree Numbers

  1. D02w.033w.100w.624w.698.268w
  2. D02w.033w.755.624w.698.268w
  3. D02w.065w.950w.681.241w
  4. D02w.092w.063w.624w.698.268w
  5. D02w.455w.426w.559w.389.703.241w

AMA Style

References

  1. National Library of Medicine. Celiprolol. Medical Subject Headings (MeSH). 2026. Unique ID D017272. http://id.nlm.nih.gov/mesh/2026/D017272
  2. Celiprolol. In: Wikipedia. https://en.wikipedia.org/wiki/Celiprolol
  3. Celiprolol. In: Wikidata. https://www.wikidata.org/wiki/Q420586
  4. Celiprolol. In: PubChem Compound. CID 2663. https://pubchem.ncbi.nlm.nih.gov/compound/2663