Chemicals and Drugs

Disintegrins

A family of polypeptides purified from snake venoms, which contain the arginine-glycine-aspartic acid (RGD) sequence. The RGD tripeptide binds to integrin receptors and thus competitively inhibits normal integrin-ligand interactions. Disintegrins thus block adhesive functions and act as platelet aggregation inhibitors.

National Library of MedicineMedical Subject Headings2026

Structured Summary

Abstract

A family of polypeptides purified from snake venoms, which contain the arginine-glycine-aspartic acid (RGD) sequence. The RGD tripeptide binds to integrin receptors and thus competitively inhibits normal integrin-ligand interactions. Disintegrins thus block adhesive functions and act as platelet aggregation inhibitors.

MeSH Record

Classification

Broader headings

Related Concepts

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Drug Class

Pharmacological Action

MeSH Record

Synonyms

1 entry terms
  • Disintegrin

MeSH Record

Aspects Covered

29 allowable subheadings

Indexed with the subheadings administration & dosage, adverse effects, agonists, analysis, antagonists & inhibitors, biosynthesis, blood, cerebrospinal fluid, chemical synthesis, chemistry, classification, deficiency, drug effects, economics, genetics, history, immunology, isolation & purification, metabolism, pharmacokinetics, pharmacology, physiology, poisoning, radiation effects, standards, supply & distribution, therapeutic use, toxicity, urine.

MeSH Record

Indexing Annotation

polypeptides from snake venom; platelet aggregation inhib

MeSH Record

History Note

97; was DISINTEGRINS (NM) 1992-96

MeSH Record

Previous Indexing

  • Peptides (1992-1996)
  • Venoms (1992-1994)

MeSH Hierarchy

Tree Number

  1. D12.644w.138

AMA Style

References

  1. National Library of Medicine. Disintegrins. Medical Subject Headings (MeSH). 2026. Unique ID D019483. http://id.nlm.nih.gov/mesh/2026/D019483
  2. Disintegrins. In: Wikidata. https://www.wikidata.org/wiki/Q41797548