Phenomena and Processes

Metabolic Inactivation

Reduction of pharmacologic activity or toxicity of a drug or other foreign substance by a living system, usually by enzymatic action. It includes those metabolic transformations that make the substance more soluble for faster renal excretion.

National Library of MedicineMedical Subject Headings2026

Structured Summary

Abstract

Reduction of pharmacologic activity or toxicity of a drug or other foreign substance by a living system, usually by enzymatic action. It includes those metabolic transformations that make the substance more soluble for faster renal excretion.

MeSH Record

Classification

Related Concepts

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MeSH Record

Synonyms

15 entry terms
  • Inactivation, Metabolic
  • Detoxication, Drug, Metabolic
  • Detoxification, Drug, Metabolic
  • Drug Detoxication, Metabolic
  • Metabolic Detoxication, Drug
  • Metabolic Detoxification, Drug
  • Metabolic Drug Inactivation
  • Detoxication, Drug Metabolic
  • Detoxication, Metabolic Drug
  • Detoxification, Drug Metabolic
  • Drug Inactivation, Metabolic
  • Drug Metabolic Detoxication
  • Drug Metabolic Detoxification
  • Inactivation, Metabolic Drug
  • Metabolic Drug Detoxication

MeSH Record

Aspects Covered

5 allowable subheadings

Indexed with the subheadings drug effects, genetics, immunology, physiology, radiation effects.

MeSH Record

Indexing Annotation

restrict to chemical changes of exogenous substances; IM general only; coordinate NIM with specific drug /pharmacokin (IM) or /metab

MeSH Record

History Note

2015 (1970); use BIOTRANSFORMATION 1970-1979

MeSH Hierarchy

Tree Numbers

MeSH Record

NLM Classification

QV 38.5

AMA Style

References

  1. National Library of Medicine. Metabolic Inactivation. Medical Subject Headings (MeSH). 2026. Unique ID D008658. http://id.nlm.nih.gov/mesh/2026/D008658
  2. Metabolic Inactivation. In: Wikidata. https://www.wikidata.org/wiki/Q70681625